"A rapid construction of 1,3,2-benzodiazaborininones [R-B(aam)] from boronic acids and anthranilamides"

作者全名："Liao, Siwei; Liu, Kai; Wu, Huili; Kuang, Qiulin; Hu, Xueyuan; Li, Yihao; Lu, Hongxiao; Yuan, Jianyong"

作者地址："[Liao, Siwei; Wu, Huili; Kuang, Qiulin; Hu, Xueyuan; Li, Yihao; Lu, Hongxiao; Yuan, Jianyong] Chongqing Med Univ, Coll Pharm, Dept Med Chem, Chongqing 400016, Peoples R China; [Liu, Kai] Chongqing Publ Hlth Med Ctr, Dept Pharm, Chongqing, Peoples R China"

通信作者："Yuan, JY (通讯作者)，Chongqing Med Univ, Coll Pharm, Dept Med Chem, Chongqing 400016, Peoples R China."

来源：RSC ADVANCES

ESI学科分类：CHEMISTRY

WOS号：WOS:000916123200001

JCR分区：Q2

影响因子：3.9

年份：2023

卷号：13

期号：4

开始页：2570

结束页：2573

文献类型：Article

关键词：　

摘要："A simple, efficient and mild methodology for the synthesis of 1,3,2-benzodiazaborininones [R-B(aam)] from boronic acids and anthranilamides on ethyl acetate is described. A series of 1,3,2-benzodiazaborininones were prepared in moderate to excellent yields at room temperature without dehydrating agents, metal catalysts, corrosive acids or other additives. Meanwhile, a multi-gram scale reaction is also performed to ensure the scalability of the reaction, and the product can be conveniently isolated by simple filtration."

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